Article, 2024

Design, Synthesis, Pharmacology, and In Silico Studies of (1S,2S,3S)-2-((S)-Amino(carboxy)methyl)-3-(carboxymethyl)cyclopropane-1-carboxylic Acid (LBG30300): A Picomolar Potency Subtype-Selective mGlu2 Receptor Agonist

JOURNAL OF MEDICINAL CHEMISTRY, ISSN 0022-2623, Volume 67, 2, Pages 1314-1326, 10.1021/acs.jmedchem.3c01811

Contributors

Liu, Na [1] Eshak, Floriane 0000-0003-2748-9398 [2] Malhaire, Fanny 0000-0001-5930-9879 [3] [4] Brabet, Isabelle [3] [4] Prezeau, Laurent [3] [4] Renard, Emma [1] Pin, Jean-Philippe 0000-0002-1423-345X [3] [4] Acher, Francine C. [2] Staudt, Markus 0000-0002-7712-1818 [1] Bunch, Lennart 0000-0002-0180-4639 (Corresponding author) [1]

Affiliations

  1. [1] Univ Copenhagen, Fac Hlth & Med Sci, Dept Drug Design & Pharmacol, DK-2100 Copenhagen OE, Denmark
    2. [NORA names: KU University of Copenhagen; University; Denmark; Europe, EU; Nordic; OECD];
  2. [2] Univ Paris Cite, SPPIN CNRS UMR 8003, Universite Paris Cite, F-75006 Paris, France
    3. [NORA names: France; Europe, EU; OECD];
  3. [3] Univ Montpellier, Inst Funct Genom, CNRS, 34094 INSERM, Montpellier, France
    4. [NORA names: France; Europe, EU; OECD];
  4. [4] Univ Montpellier, Inst Funct Genom, CNRS, 34094 INSERM, Montpellier, France
    5. [NORA names: France; Europe, EU; OECD]

Abstract

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